Browse by Basel Contributors ID
2016Kleeb, Simon and Jiang, Xiaohua and Frei, Priska and Sigl, Anja and Bezençon, Jacqueline and Bamberger, Karen and Schwardt, Oliver and Ernst, Beat. (2016) FimH Antagonists: Phosphate Prodrugs Improve Oral Bioavailability. Journal of Medicinal Chemistry, 59 (7). pp. 3163-3182. Eris, Deniz and Preston, Roland C. and Scharenberg, Meike and Hulliger, Fabian and Abgottspon, Daniela and Pang, Lijuan and Jiang, Xiaohua and Schwardt, Oliver and Ernst, Beat. (2016) The Conformational Variability of FimH: Which Conformation Represents the Therapeutic Target? ChemBioChem, 17 (11). pp. 1012-1020. 2015Kleeb, Simon and Pang, Lijuan and Mayer, Katharina and Eris, Deniz and Sigl, Anja and Preston, Roland C. and Zihlmann, Pascal and Sharpe, Timothy and Jakob, Roman P. and Abgottspon, Daniela and Hutter, Aline S. and Scharenberg, Meike and Jiang, Xiaohua and Navarra, Giulio and Rabbani, Said and Smiesko, Martin and Lüdin, Nathalie and Bezençon, Jacqueline and Schwardt, Oliver and Maier, Timm and Ernst, Beat. (2015) FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile. Journal of Medicinal Chemistry, 58 (5). pp. 2221-2239. Fiege, Brigitte and Rabbani, Said and Preston, Roland C. and Jakob, Roman P. and Zihlmann, Pascal and Schwardt, Oliver and Jiang, Xiaohua and Maier, Timm and Ernst, Beat. (2015) The Tyrosine Gate of the Bacterial Lectin FimH : a Conformational Analysis by NMR Spectroscopy and X-ray Crystallography. ChemBioChem, 16 (8). pp. 1235-1246. 2013Scharenberg, Meike and Jiang, Xiaohua and Pang, Lijuan and Navarra, Giulio and Rabbani, Said and Binder, Florian and Schwardt, Oliver and Ernst, Beat. (2013) Kinetic properties of carbohydrate–lectin interactions: FimH antagonists. ChemMedChem, 9 (1). pp. 78-83. 2012Jiang, Xiaohua and Abgottspon, Daniela and Kleeb, Simon and Rabbani, Said and Scharenberg, Meike and Wittwer, Matthias and Haug, Martina and Schwardt, Oliver and Ernst, Beat. (2012) Anti-adhesion therapy for urinary tract infections - a balanced PK/PD-profile proved to be key for success. Journal of Medicinal Chemistry, 55 (10). pp. 4700-4713. 2011Scharenberg, Meike and Abgottspon, Daniela and Cicek, Evelin and Jiang, Xiaohua and Schwardt, Oliver and Rabbani, Said and Ernst, Beat. (2011) A Flow Cytometry-based Assay for Screening FimH Antagonists. Assay and Drug Development Technologies, 9 (5). pp. 455-464. |